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Investigational noncardiovascular uses of phosphodiesterase-5 inhibitors.

Authors: Robert A Kloner|||Gary Comstock|||Laurence A Levine|||Steven Tiger|||Vera J Stecher

Journal: Expert opinion on pharmacotherapy

Publication Type: Journal Article

Date: 2011

DOI: 10.1517/14656566.2011.600306

ID: 21774742

Affiliations:

Affiliations

    The Heart Institute, Good Samaritan Hospital, 1225 Wilshire Blvd, Los Angeles, CA 90017-2395, USA. rkloner@goodsam.org||||||||||||

Abstract

At the present time, inhibitors of phosphodiesterase type 5 (PDE5) have Food and Drug Administration approval only for the treatment of erectile dysfunction and pulmonary artery hypertension, for which their mechanism of action is vasodilation and augmentation of blood flow by impeding PDE5-mediated breakdown of cyclic guanosine monophosphate. However, these agents are also being investigated in a wide range of other potential medical and surgical applications for which current treatment options are limited and in which their mechanism of action may be the same as or different from their effects in the two approved indications. Even if only some of these potential applications prove useful, the effect on clinical practice could be far reaching.


Chemical List

    Phosphodiesterase 5 Inhibitors